Developer · United States
Intra-Cellular Therapies, Inc.
A biopharmaceutical company focused on the development and commercialization of therapeutics for central nervous system disorders; developer of CAPLYTA (lumateperone). Acquired by Johnson & Johnson in April 2025 and now operated as part of Johnson & Johnson Innovative Medicine.
Pipeline (3)
- SchizophreniaApprovedApproved
- Major depressive disorderApprovedApproved
- Bipolar depressionApprovedApproved
- Bipolar disorderPhase 3Recruiting
- Autism spectrum disorderPhase 3Recruiting
- Alzheimer's diseasePhase 2Recruiting
- Generalized anxiety disorderPhase 2Recruiting
- Agitation in Alzheimer's diseasePhase 2Recruiting
- Parkinson's diseasePhase 2Active
Deals & partnerships
- ITI-1284 (deulumateperone)Led by Johnson & Johnson
- Lenrispodun (ITI-214)Led by Johnson & Johnson
- Lumateperone (ITI-007)Led by Johnson & JohnsonLicensor Bristol-Myers Squibb Company
- Apr 2, 2025AcquisitionJohnson & Johnson acquires Intra-Cellular TherapiesJohnson & Johnson completed its acquisition of Intra-Cellular Therapies for $132.00 per share in cash (~$14.6B), closing April 2, 2025. ITCI delisted from NASDAQ and became a unit within Johnson & Johnson Innovative Medicine. Adds CAPLYTA (lumateperone) and the pipeline (ITI-1284, lenrispodun).
- May 2005Licensing dealIntra-Cellular in-licenses lumateperone (ITI-007) from Bristol-Myers SquibbIntra-Cellular Therapies obtained an exclusive, worldwide license to lumateperone (ITI-007) and related CNS compounds from Bristol-Myers Squibb in 2005, the basis for its worldwide rights to CAPLYTA.
Catalysts · 9 upcoming · 8 reported
- 2025Delayed
Lenrispodun (ITI-214)forParkinson's diseaseTopline data
Phase 2 ITI-214-202 topline in Parkinson's disease (lenrispodun 30 mg vs placebo, Hauser-diary primary at Day 29).
- 1H 2026Anticipated
Lumateperone (ITI-007)forBipolar disorderTopline data
Anticipated topline from Phase 3 Study 451 (NCT06462586) of lumateperone 42 mg in acute bipolar mania (YMRS at Week 3).
- 2H 2026Anticipated
Lumateperone (ITI-007)forBipolar disorderTopline data
Anticipated topline from Phase 3 Study 452 (NCT06462612) of lumateperone 42 mg in acute bipolar mania (YMRS at Week 3).
- 1H 2027Anticipated
Lumateperone (ITI-007)forAutism spectrum disorderTopline data
Anticipated topline of Study 602, the second pivotal Phase 3 of lumateperone for irritability associated with autism spectrum disorder (pediatric); primary endpoint ABC-Irritability at Week 6.
- 1H 2027Anticipated
Lumateperone (ITI-007)forAutism spectrum disorderTopline data
Anticipated topline of Study 601, the first pivotal Phase 3 of lumateperone for irritability associated with autism spectrum disorder (pediatric); primary endpoint ABC-Irritability at Week 6.
- Mid-2027Anticipated
ITI-1284 (deulumateperone)forGeneralized anxiety disorderTopline data
Anticipated Phase 2 topline for monotherapy ITI-1284 in GAD (NCT06701903); primary completion targeted June 2027.
- Mid-2027Anticipated
ITI-1284 (deulumateperone)forGeneralized anxiety disorderTopline data
Anticipated Phase 2 topline for adjunctive ITI-1284 in GAD (NCT06480383); primary completion targeted June 2027.
- 2H 2027Anticipated
ITI-1284 (deulumateperone)forAlzheimer's diseaseTopline data
Anticipated Phase 2 topline for ITI-1284 in psychosis associated with Alzheimer's disease (NCT06540833); primary completion targeted September 2027.
- Q4 2027Anticipated
ITI-1284 (deulumateperone)forAgitation in Alzheimer's diseaseTopline data
Anticipated Phase 2 topline for ITI-1284 in agitation associated with Alzheimer's dementia (NCT06651567); primary completion targeted October 2027.
Recently reported
- 2026-04-27met
Lumateperone (ITI-007)forSchizophreniaRegulatory
FDA approved Caplyta (lumateperone) sNDA adding relapse-prevention data in schizophrenia (Study 304: HR 0.37, 63% lower relapse risk, p=0.0002).
- 2025-11-06met
Lumateperone (ITI-007)forMajor depressive disorderRegulatory
FDA approved Caplyta (lumateperone) as adjunctive therapy with antidepressants for MDD in adults.
- 2024-06-18met
Lumateperone (ITI-007)forMajor depressive disorderTopline data
Study 502 positive: lumateperone + antidepressant met MADRS primary (-4.5 vs placebo, p<0.0001) and CGI-S key secondary at Week 6.
- 2024-04-16met
Lumateperone (ITI-007)forMajor depressive disorderTopline data
Study 501 positive: lumateperone + antidepressant met MADRS primary (-4.9 vs placebo, p<0.0001) and CGI-S key secondary at Week 6.
- 2023-02-13met
Lumateperone (ITI-007)forBipolar depressionFull results
Study 402 positive (42 mg): lumateperone adjunctive to lithium/valproate met the MADRS Week-6 primary in bipolar depression (LSMD -2.4, p=0.02).
- 2021-12-20met
Lumateperone (ITI-007)forBipolar depressionRegulatory
FDA approved Caplyta (lumateperone) for bipolar I and II depression in adults, as monotherapy and as adjunctive therapy with lithium or valproate.
- 2021-09-23met
Lumateperone (ITI-007)forBipolar depressionFull results
Study 404 positive: lumateperone 42 mg monotherapy met the MADRS Week-6 primary in bipolar I/II depression (LSMD -4.6, ES -0.56, p<0.0001).
- 2019-12-20met
Lumateperone (ITI-007)forSchizophreniaRegulatory
FDA approved Caplyta (lumateperone) 42 mg once daily for the treatment of schizophrenia in adults.
Recent activity
- Apr 27, 2026ReadoutLumateperone (ITI-007)·SchizophreniametFDA approved Caplyta (lumateperone) sNDA adding relapse-prevention data in schizophrenia (Study 304: HR 0.37, 63% lower relapse risk, p=0.0002).source ↗
- Nov 6, 2025ReadoutLumateperone (ITI-007)·Major depressive disordermetFDA approved Caplyta (lumateperone) as adjunctive therapy with antidepressants for MDD in adults.source ↗
- Nov 4, 2025Phase changeLenrispodun (ITI-214)·Parkinson's diseasePhase 2Phase 2 ITI-214-202 reached final completion (primary completion 2025-10-28); 79 patients enrolled. Registry status COMPLETED as of last update 2026-05-22. No topline results disclosed yet.source ↗
- Feb 21, 2025Phase changeITI-1284 (deulumateperone)·Agitation in Alzheimer's diseasePhase 2Intra-Cellular Therapies FY2024 corporate update reports patient enrollment ongoing in the Phase 2 program evaluating ITI-1284 in agitation associated with Alzheimer's disease (alongside the Phase 2 Alzheimer's psychosis program).source ↗
- Feb 21, 2025Phase changeLumateperone (ITI-007)·Autism spectrum disorderPhase 3Intra-Cellular Therapies FY2024 corporate update: 'in the fourth quarter of 2024, we commenced patient enrollment in two Phase 3 studies in pediatric patients for the treatment of irritability associated with autism spectrum disorder' (Studies 601/602; NCT06690398, NCT06706674).source ↗
- Dec 3, 2024Phase changeLumateperone (ITI-007)·Major depressive disorderFiled (NDA)Intra-Cellular Therapies submitted the sNDA to FDA for Caplyta (lumateperone) as adjunctive therapy for MDD, based on Studies 501 and 502.source ↗
- Nov 22, 2024Phase changeLumateperone (ITI-007)·Autism spectrum disorderPhase 3Study 601 (NCT06690398, ITI-007-601) Phase 3 in pediatric irritability associated with autism spectrum disorder started; randomized, double-blind, placebo-controlled, n=174, primary endpoint ABC-Irritability at Week 6. Study start date per ClinicalTrials.gov.source ↗
- Nov 21, 2024Phase changeITI-1284 (deulumateperone)·Generalized anxiety disorderPhase 2Second GAD trial started: monotherapy Phase 2 study NCT06701903 (ITI-1284 10 mg / 20 mg sublingual vs placebo, n~570).source ↗
- Oct 22, 2024Phase changeITI-1284 (deulumateperone)·Agitation in Alzheimer's diseasePhase 2Phase 2 agitation-in-Alzheimer's-dementia trial started: NCT06651567 (ITI-1284 10-20 mg sublingual ODT once daily vs placebo, flexible-dose, n~320; primary endpoint CMAI total score at Week 12). Actual study start per ClinicalTrials.gov.source ↗
- Aug 15, 2024Phase changeITI-1284 (deulumateperone)·Alzheimer's diseasePhase 2Phase 2 Alzheimer's-disease psychosis trial started: NCT06540833, a multicenter, randomized, double-blind, placebo-controlled, flexible-dose study of ITI-1284 10 mg / 20 mg once-daily sublingual ODT vs placebo (n=370), 6-week treatment, primary outcome BEHAVE-AD psychosis subscale at Week 6.source ↗
- Aug 5, 2024Phase changeITI-1284 (deulumateperone)·Generalized anxiety disorderPhase 2First GAD trial started: adjunctive Phase 2 study NCT06480383 (ITI-1284 10 mg / 20 mg sublingual vs placebo in patients with inadequate response to GAD treatment, n~705).source ↗
- Jul 17, 2024Phase changeLumateperone (ITI-007)·Bipolar disorderPhase 3Study 452 (NCT06462612, ITI-007-452) started — second Phase 3 acute bipolar-mania study, same design (lumateperone 42 mg vs placebo, 3-week, YMRS Week 3 primary). CT.gov start date 17 Jul 2024; status RECRUITING. Together the two studies form the pivotal acute-mania package. Intra-Cellular reported both were initiated in Q2 2024 with enrollment ongoing.source ↗
Trials recruiting · 10 recruiting of 22 sponsored
- Phase 3Lumateperone (ITI-007)
Study 602: A Randomized, Double-blind, Placebo-controlled, Multicenter Study to Assess the Efficacy and Safety of Lumateperone in the Treatment of Irritability Associated With Autism Spectrum Disorder in Pediatric Patients 5 to 17 Years of Age
- Phase 3Lumateperone (ITI-007)
Study 601: A Randomized, Double-blind, Placebo-controlled, Multicenter Study to Assess the Efficacy and Safety of Lumateperone in the Treatment of Irritability Associated With Autism Spectrum Disorder in Pediatric Patients 5 to 17 Years of Age
- Phase 3Lumateperone (ITI-007)
Study 452: A Multicenter, Randomized, Double-blind, Placebo-controlled Study to Assess the Efficacy and Safety of Lumateperone in the Acute Treatment of Patients With Manic Episodes or Manic Episodes With Mixed Features Associated With Bipolar I Disorder (Bipolar Mania)
- Phase 3Lumateperone (ITI-007)
Study 451: A Multicenter, Randomized, Double-blind, Placebo-controlled Study to Assess the Efficacy and Safety of Lumateperone in the Acute Treatment of Patients With Manic Episodes or Manic Episodes With Mixed Features Associated With Bipolar I Disorder (Bipolar Mania)
- Phase 3Lumateperone (ITI-007)
An Open-label, Multicenter Trial to Assess the Safety and Tolerability of Lumateperone in the Treatment of Pediatric Patients With Schizophrenia, Bipolar Disorder or Autism Spectrum Disorder
- Phase 3Lumateperone (ITI-007)
Study 505: A Randomized, Double-Blind, Placebo-controlled Multicenter Study to Assess the Efficacy and Safety of Lumateperone as Adjunctive Therapy in the Treatment of Patients With Major Depressive Disorder
- Phase 2ITI-1284 (deulumateperone)
A Multicenter, Randomized, Double-blind, Placebo-controlled Study to Assess the Efficacy, Safety, and Tolerability of ITI-1284 as Monotherapy Treatment in Patients With Generalized Anxiety Disorder
- Phase 2ITI-1284 (deulumateperone)
A Multicenter, Randomized, Double-blind, Placebo-controlled, Flexible-dose Study of the Efficacy, Safety, and Tolerability of ITI-1284 in Patients With Agitation Associated With Alzheimer's Dementia
- Phase 2ITI-1284 (deulumateperone)
A Multicenter, Randomized, Double-blind, Placebo-controlled, Flexible-dose Study to Assess the Efficacy, Safety, and Tolerability of ITI-1284 in Patients With Psychosis Associated With Alzheimer's Disease
- Phase 2ITI-1284 (deulumateperone)
A Multicenter, Randomized, Double-blind, Placebo-controlled Study to Assess the Efficacy, Safety, and Tolerability of ITI-1284 as an Adjunctive Treatment in Patients With Generalized Anxiety Disorder Who Have an Inadequate Response to Generalized Anxiety Disorder Treatment
Competitive landscape
Other companies developing against Intra-Cellular Therapies, Inc.'s targets or indications.
- Definium Therapeutics, Inc.2 compounds5-HT2AGeneralized anxiety disorderMajor depressive disorderAutism spectrum disorder
- Vanda Pharmaceuticals Inc.2 compounds5-HT2ASchizophreniaMajor depressive disorderBipolar disorder
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- Autobahn Therapeutics, Inc.1 compoundMajor depressive disorderBipolar depression
- Axsome Therapeutics, Inc.2 compoundsAgitation in Alzheimer's diseaseMajor depressive disorder
- Beckley Psytech Limited1 compound5-HT2AMajor depressive disorder
- BioXcel Therapeutics, Inc.1 compoundAgitation in Alzheimer's diseaseSchizophrenia