Drug target · SLC1A2

EAAT2

Excitatory amino acid transporter 2 (glial high-affinity glutamate transporter, GLT-1)

1 compound in the CNS pipeline acts on EAAT2.

Compounds targeting EAAT2

CompoundActionAffinityLead programDeveloper
Troriluzole (BHV-4157)primarySmall moleculeModulatorDiscontinuedObsessive-compulsive disorderBiohaven Ltd.