Drug target · DRD5
D5 receptor
Dopamine D5 receptor
2 compounds in the CNS pipeline act on D5 receptor.
Compounds targeting D5 receptor
| Compound | Action | Affinity | Lead program | Developer |
|---|---|---|---|---|
| EcopipamSmall molecule | Antagonist | pKi 8.3 | Filed (NDA)Tourette syndrome | Emalex Biosciences Inc. |
| TavapadonSmall molecule | Partial agonist | Ki 13 nM | Filed (NDA)Parkinson's disease | Cerevel Therapeutics Holdings, Inc. |