Drug target · DRD1

D1 receptor

Dopamine D1 receptor

2 compounds in the CNS pipeline act on D1 receptor.

Compounds targeting D1 receptor

CompoundActionAffinityLead programDeveloper
EcopipamprimarySmall moleculeAntagonistpKi 8.3Filed (NDA)Tourette syndromeEmalex Biosciences Inc.
TavapadonprimarySmall moleculePartial agonistKi 9 nMFiled (NDA)Parkinson's diseaseCerevel Therapeutics Holdings, Inc.