Drug target · SLC6A2

Norepinephrine transporter (NET)

Sodium-dependent noradrenaline transporter

2 compounds in the CNS pipeline act on Norepinephrine transporter (NET).

Compounds targeting Norepinephrine transporter (NET)

CompoundActionAffinityLead programDeveloper
AXS-05 (dextromethorphan-bupropion)Small moleculeReuptake inhibitorApprovedAgitation in Alzheimer's diseaseAxsome Therapeutics, Inc.
Ammoxetine (S-071031B)Small moleculeInhibitorPhase 3Major depressive disorderCSPC ZhongQi Pharmaceutical Technology (Shijiazhuang) Co., Ltd.