Drug target · OPRM1
mu-opioid receptor
mu-type opioid receptor (MOP)
1 compound in the CNS pipeline acts on mu-opioid receptor.
Compounds targeting mu-opioid receptor
| Compound | Action | Affinity | Lead program | Developer |
|---|---|---|---|---|
| LYBALVI (olanzapine/samidorphan)Small molecule | Antagonist | Ki 0.05 nM | Phase 3Schizophrenia | Alkermes plc |