Drug target · GRM3

mGlu3

Metabotropic glutamate receptor 3

2 compounds in the CNS pipeline act on mGlu3.

Compounds targeting mGlu3

CompoundActionAffinityLead programDeveloper
Pomaglumetad methionilSmall moleculeAgonistKi 92 nMDiscontinuedSchizophreniaEli Lilly and Company
TS-161Small moleculeAntagonistKi 2.83 nMDiscontinuedTreatment-resistant depressionTaisho Pharmaceutical Co., Ltd.