Drug target · NR3C1

Glucocorticoid receptor

Glucocorticoid receptor (nuclear receptor subfamily 3 group C member 1)

1 compound in the CNS pipeline acts on Glucocorticoid receptor.

Compounds targeting Glucocorticoid receptor

CompoundActionAffinityLead programDeveloper
PT150 (Org 34517)primarySmall moleculeAntagonist—Phase 2Post-traumatic stress disorderMerck & Co., Inc.