Drug target · GABRA5
GABA-A receptor alpha-5
Gamma-aminobutyric acid type A receptor subunit alpha-5
1 compound in the CNS pipeline acts on GABA-A receptor alpha-5.
Compounds targeting GABA-A receptor alpha-5
| Compound | Action | Affinity | Lead program | Developer |
|---|---|---|---|---|
| Darigabat (CVL-865)Small molecule | PAM | Ki 18 nM | DiscontinuedEpilepsy | Cerevel Therapeutics Holdings, Inc. |