Drug target · GABRA3
GABA-A receptor alpha-3
Gamma-aminobutyric acid type A receptor subunit alpha-3
1 compound in the CNS pipeline acts on GABA-A receptor alpha-3.
Compounds targeting GABA-A receptor alpha-3
| Compound | Action | Affinity | Lead program | Developer |
|---|---|---|---|---|
| Darigabat (CVL-865)Small molecule | PAM | Ki 1.1 nM | DiscontinuedEpilepsy | Cerevel Therapeutics Holdings, Inc. |