Drug target · ADRA2C
alpha-2C adrenoceptor
Alpha-2C adrenergic receptor
1 compound in the CNS pipeline acts on alpha-2C adrenoceptor.
Compounds targeting alpha-2C adrenoceptor
| Compound | Action | Affinity | Lead program | Developer |
|---|---|---|---|---|
| Dexmedetomidine sublingual film (BXCL501)Small molecule | Agonist | — | Phase 1/2Opioid use disorder | BioXcel Therapeutics, Inc. |