Drug target · ADRA2C

alpha-2C adrenoceptor

Alpha-2C adrenergic receptor

1 compound in the CNS pipeline acts on alpha-2C adrenoceptor.

Compounds targeting alpha-2C adrenoceptor

CompoundActionAffinityLead programDeveloper
Dexmedetomidine sublingual film (BXCL501)Small moleculeAgonistPhase 3Agitation in Alzheimer's diseaseBioXcel Therapeutics, Inc.