Drug target · ADRA2B

alpha-2B adrenoceptor

Alpha-2B adrenergic receptor

1 compound in the CNS pipeline acts on alpha-2B adrenoceptor.

Compounds targeting alpha-2B adrenoceptor

CompoundActionAffinityLead programDeveloper
Dexmedetomidine sublingual film (BXCL501)Small moleculeAgonistPhase 3Agitation in Alzheimer's diseaseBioXcel Therapeutics, Inc.