Drug target · ADRA2A

alpha-2A adrenoceptor

Alpha-2A adrenergic receptor

1 compound in the CNS pipeline acts on alpha-2A adrenoceptor.

Compounds targeting alpha-2A adrenoceptor

CompoundActionAffinityLead programDeveloper
Dexmedetomidine sublingual film (BXCL501)primarySmall moleculeAgonistFiled (NDA)SchizophreniaBioXcel Therapeutics, Inc.