Drug target · ADORA2A
Adenosine A2A receptor
Adenosine A2A receptor
1 compound in the CNS pipeline acts on Adenosine A2A receptor.
Compounds targeting Adenosine A2A receptor
| Compound | Action | Affinity | Lead program | Developer |
|---|---|---|---|---|
| SipagladenantprimarySmall molecule | Inverse agonist | pKi 9.93 | DiscontinuedParkinson's disease | Kyowa Kirin Co., Ltd. |